Wednesday 7 July 2021

Zuclopenthixol

Carisbamate:

Carisbamate yog kev sim tshuaj anticonvulsant uas tau tsim kho los ntawm Johnson & Johnson Pharmaceutical Kev Tshawb Fawb thiab Kev Txhim Kho tab sis tsis tau muag khoom.

Retigabine:

Retigabine (INN) lossis ezogabine (USAN) yog cov tshuaj anticonvulsant siv los ua kev kho mob rau cov mob vwm feem ib feem hauv kev kho mob-laus tus neeg mob. Cov tshuaj tau txhim kho los ntawm Valeant Pharmaceuticals thiab GlaxoSmithKline. Nws tau pom zoo los ntawm European Medicines Agency nyob rau hauv lub npe kev lag luam Trobalt thaum Lub Peb Hlis 28, 2011, thiab los ntawm Tsoom Fwv Tswj Khoom Noj thiab Tshuaj (FDA), nyob hauv kev lag luam npe Potiga , thaum Lub Rau Hli 10, 2011. Cov khoom lag luam tau raug txiav tawm thaum Lub Rau Hli Xyoo 2017.

Perampanel:

Perampanel , muag nyob hauv cov npe lag luam lub npe Fycompa , yog ib qho tshuaj tiv thaiv kev puas ntsoog uas tsim los ntawm Eisai Co. uas yog siv ntxiv rau lwm cov tshuaj los kho kho mob ib nrab thiab feem ntau tonic-clonic qaug dab peg rau cov neeg laus dua kaum ob xyoos. Nws tau pom zoo thawj zaug hauv xyoo 2012, thiab txog xyoo 2016, nws lub luag haujlwm tseem ceeb hauv kev kho tus mob ntsig txog kabmob mus rau lwm cov tshuaj tsis pom tseeb. Nws yog thawj cov tshuaj tua kab mob hauv chav kawm ntawm cov xaiv tshuaj uas tsis muaj kev sib tw ntawm cov tshuaj tiv thaiv AMPA.

Beclamide:

Beclamide yog ib qho tshuaj uas muaj cov tshuaj tiv thaiv anticonvulsant. Nws yog tsis siv.

ATC code N04:

ATC code N04 Cov tshuaj tiv thaiv cov tshuaj tiv thaiv kab mob yog kev siv tshuaj ntawm Anatomical Kev Ntsuas Tshuaj Classification System, ib qho kev hloov kho cov txheej txheem alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N04 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

ATC code N04:

ATC code N04 Cov tshuaj tiv thaiv cov tshuaj tiv thaiv kab mob yog kev siv tshuaj ntawm Anatomical Kev Ntsuas Tshuaj Classification System, ib qho kev hloov kho cov txheej txheem alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N04 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

ATC code N04:

ATC code N04 Cov tshuaj tiv thaiv cov tshuaj tiv thaiv kab mob yog kev siv tshuaj ntawm Anatomical Kev Ntsuas Tshuaj Classification System, ib qho kev hloov kho cov txheej txheem alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N04 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

Trihexyphenidyl:

Trihexyphenidyl , aka tseem hu ua benzhexol , trihex , lossis txawm THP yog tus kabmob antiparkinsonian ntawm chav kawm antimuscarinic. Nws tau pom zoo los ntawm FDA rau kev kho mob ntawm Parkinson xyoo 2003.

Biperiden:

Biperiden , muag nyob hauv hom tshuaj npe Akineton ntawm lwm tus, yog cov tshuaj siv los kho tus kab mob Parkinson thiab qee yam tshuaj ua kom lub zog txav tsis zoo. Nws tsis pom zoo rau qhov ua tuaj ntawm qhov nqua tuaj. Nws yog noj ntawm qhov ncauj, txhaj rau hauv leeg ntshav, lossis leeg leeg.

Metixene:

Metixene , tseem hu ua methixene , yog anticholinergic siv los ua Kev tswj hwm ntawm Parkinson tus kab mob # Tshuaj kho mob} antiparkinsonian tus neeg sawv cev.

Procyclidine:

Procyclidine yog cov tshuaj anticholinergic feem ntau siv rau kev kho mob los ntawm kev quav yeeb tshuaj parkinsonism, akathisia thiab mob dystonia mob siab; Kab mob Parkinson; thiab idiopathic los yog theem nrab dystonia.

Profenamine:

Profenamine yog ib qho phenothiazine derivative siv los ua tus neeg sawv cev antiparkinsonian uas muaj anticholinergic, antihistamine, thiab antiadrenergic kev ua. Nws kuj tseem raug siv rau hauv kev txo qis ntawm qhov mob ua ke (extrapyramidal syndrome) los ntawm cov tshuaj xws li lwm cov phenothiazine tebchaw, tab sis, zoo li lwm cov khoom sib txuas nrog cov khoom antimuscarinic, tsis muaj txiaj ntsig tawm ntawm tardive dyskinesia.

Dexetimide:

Dexetimide yog piperidine anticholinergic. Nws yog cov muscarinic antagonist uas yog siv los kho kev quav yeeb tshuaj parkinsonism. Dexetimide nrhiav tau ntawm Janssen Pharmaceutica hauv xyoo 1968.

Phenglutarimide:

Phenglutarimide yog tshuaj tua kabmob (anticholinergic) siv los ua tus kabmob antiparkinsonian.

Mazaticol:

Mazaticol ( Pentona ) yog ib qho anticholinergic siv los ua tus sawv cev tshuaj tua kab mob rau hauv Nyij Pooj.

Bornaprine:

Bornaprine yog cov tshuaj tua kab mob anticholinergic uas feem ntau siv los kho tus mob Parkinson. Tsis tas li ntawd, bornaprine tau siv los kho lwm yam cuam tshuam, suav nrog hyperhidrosis.

Tropatepine:

Tropatepine yog ib qho tshuaj anticholinergic siv los ua tus sawv cev rau tshuaj tua kabmob.

ATC code N04:

ATC code N04 Cov tshuaj tiv thaiv cov tshuaj tiv thaiv kab mob yog kev siv tshuaj ntawm Anatomical Kev Ntsuas Tshuaj Classification System, ib qho kev hloov kho cov txheej txheem alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N04 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

Etanautine:

Etanautine , tseem hu ua diphenhydramine monoacefyllinate , yog anticholinergic siv los ua tus sawv cev antiparkinsonian. Nws yog 1: 1 ntsev ntawm diphenhydramine nrog acefylline, zoo ib yam li diphenhydramine / 8-chlorotheophylline ua ke cov khoom lag luam dimenhydrinate.

Orphenadrine:

Orphenadrine yog ib qho tshuaj anticholinergic ntawm ethanolamine antihistamine chav kawm; Nws yog ze rau ntawm diphenhydramine. Nws yog siv los kho cov leeg mob thiab los pab tswj lub cev muaj zog hauv Parkinson tus kab mob, tab sis tau siv tshuaj ntau dua los hloov cov tshuaj tshiab. Qhov tshuaj yeeb dej caw no yog tshuaj yeeb tshuaj vim nws muaj ntau cov txheej txheem ntawm kev coj ua hauv kev sib txawv. Nws tau tshawb pom thiab tsim tawm xyoo 1940s.

ATC code N04:

ATC code N04 Cov tshuaj tiv thaiv cov tshuaj tiv thaiv kab mob yog kev siv tshuaj ntawm Anatomical Kev Ntsuas Tshuaj Classification System, ib qho kev hloov kho cov txheej txheem alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N04 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

Benzatropine:

Benzatropine (INN), lub npe hu ua benztropine hauv Tebchaws Asmeskas thiab Nyijpooj, yog cov tshuaj siv los kho hom mob qoj ib ce vim muaj cov tshuaj tiv thaiv kab mob hu ua dystonia thiab parkinsonism. Nws tsis muaj txiaj ntsig rau tardive dyskinesia. Nws noj ntawm qhov ncauj lossis los ntawm txhaj tshuaj rau hauv leeg ntshav lossis leeg leeg. Cov txiaj ntsig tau pom hauv ob teev thiab kav ntev txog li kaum teev.

Etybenzatropine:

Etybenzatropine (INN), tseem hu ua ethybenztropine thiab tropethydrylin , yog anticholinergic / antihistamine ua lag luam nyob hauv kev lag luam tawm npe Panolid , Ponalid , thiab Ponalide , uas yog siv los ua tus sawv cev tiv thaiv kabmob. Zoo li nws cov analogue benzatropine, nws tuaj yeem ua raws li dopamine reuptake inhibitor.

ATC code N04:

ATC code N04 Cov tshuaj tiv thaiv cov tshuaj tiv thaiv kab mob yog kev siv tshuaj ntawm Anatomical Kev Ntsuas Tshuaj Classification System, ib qho kev hloov kho cov txheej txheem alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N04 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

ATC code N04:

ATC code N04 Cov tshuaj tiv thaiv cov tshuaj tiv thaiv kab mob yog kev siv tshuaj ntawm Anatomical Kev Ntsuas Tshuaj Classification System, ib qho kev hloov kho cov txheej txheem alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N04 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

L-DOPA:

l -DOPA , tseem hu ua levodopa thiab l -3,4-dihydroxyphenylalanine , yog cov amino acid uas tau tsim thiab siv ua ib feem ntawm kev ib txwm muaj tsiaj txhu tib neeg, nrog rau qee yam tsiaj thiab nroj tsuag. Tib neeg, nrog rau ib feem ntawm lwm yam tsiaj uas siv l -DOPA hauv lawv cov tsiaj txhu, ua nws ntawm biosynthesis los ntawm cov amino acid l -tyrosine . l -DOPA yog qhov kev qhia ua ntej rau cov neurotransmitters dopamine, norepinephrine (noradrenaline), thiab epinephrine (adrenaline), uas tau paub zoo ua catecholamines. Tsis tas li ntawd, l -DOPA nws tus kheej daws cov teeb meem neurotrophic tso tawm los ntawm lub hlwb thiab CNS. l -DOPA tuaj yeem tsim tawm thiab hauv nws daim ntawv dawb huv yog muag raws li cov tshuaj psychoactive nrog INN levodopa; cov npe lag luam suav nrog Sinemet, Pharmacopa, Atamet, thiab Stalevo. Raws li cov tshuaj, nws yog siv nyob rau hauv kev kho mob chaw kho mob ntawm Parkinson tus kab mob thiab dopamine-teb dystonia.

Melevodopa:

Melevodopa yog ib tus neeg sawv cev rau dopaminergic. Nws yog cov methyl ester ntawm levodopa. Nws siv nyob rau hauv daim ntawv ntsiav tshuaj raws li ib qho effervescent prodrug nrog 250 lub sijhawm dej solubility ntawm ntsiav tshuaj levodopa.

ATC code N04:

ATC code N04 Cov tshuaj tiv thaiv cov tshuaj tiv thaiv kab mob yog kev siv tshuaj ntawm Anatomical Kev Ntsuas Tshuaj Classification System, ib qho kev hloov kho cov txheej txheem alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N04 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

Amantadine:

Amantadine , muag nyob rau hauv cov npe lag luam Gocovri ntawm lwm tus, yog cov tshuaj siv los kho dyskinesia cuam tshuam nrog parkinsonism thiab mob khaub thuas tshwm sim los ntawm hom A influenzavirus, txawm hais tias nws siv rau tom kawg tsis pom zoo vim muaj ntau yam tshuaj tiv thaiv. Nws ua raws li nicotinic antagonist, dopamine agonist, thiab tsis yooj yim NMDA antagonist. Antiviral mechanism ntawm kev ua yog antagonism ntawm lub influenzavirus A M2 proton channel, uas tiv thaiv kev tiv thaiv kev ua kom mob siab.

ATC code N04:

ATC code N04 Cov tshuaj tiv thaiv cov tshuaj tiv thaiv kab mob yog kev siv tshuaj ntawm Anatomical Kev Ntsuas Tshuaj Classification System, ib qho kev hloov kho cov txheej txheem alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N04 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

Bromocriptine:

Bromocriptine , thaum xub thawj ua lag luam yog Parlodel thiab tom qab ntawd muaj ntau lub npe lag luam, yog ergoline derivative thiab dopamine agonist uas tau siv rau kev kho mob qog nqaij hlav, Parkinson tus kab mob, hyperprolactinaemia, neuroleptic malignant syndrome, thiab, raws li qhov txuas, mob ntshav qab zib hom 2.

Pergolide:

Pergolide , muag nyob rau hauv cov npe lag luam Permax thiab Prascend (kws kho tsiaj) nrog lwm tus, yog ergoline-based dopamine receptor agonist siv nyob rau qee lub tebchaws rau kev kho mob Parkinson. Tus kab mob Parkinson tau cuam tshuam nrog kev txo qis dopamine kev ua si hauv qhov muaj nuj nqis ntawm lub hlwb. Pergolide ua rau ntau ntawm tib lub receptors li dopamine kom nce kev ua si.

Dihydroergocryptine:

Dihydroergocryptine ( DHEC ), muag nyob hauv cov lag luam muaj npe Almirid thiab Cripar ntawm lwm tus, yog dopamine agonist ntawm pawg ergoline uas tau siv los ua tus sawv cev antiparkinson hauv kev kho mob ntawm Parkinson tus kab mob. Nws yog noj ntawm qhov ncauj.

Ropinirole:

Ropinirole , muag nyob rau hauv hom tshuaj npe hu ua Requip ntawm lwm tus, yog cov tshuaj siv los kho tus kab mob Parkinson (PD) thiab mob ceg tsis tswm (RLS). Hauv PD qhov tshuaj xav tau kho kom haum rau cov nyhuv thiab kev kho mob yuav tsum tsis txhob tsum sai. Nws yog noj ntawm qhov ncauj.

Pramipexole:

Pramipexole , muag nyob hauv cov lag luam muaj npe Mirapex ntawm lwm tus, yog cov tshuaj siv los kho Parkinson tus kab mob (PD) thiab mob ceg tsis tswm (RLS). Hauv Parkinson tus kab mob nws yuav siv ib leeg los yog ua ke nrog levodopa. Nws yog noj ntawm qhov ncauj. Pramipexole yog dopamine agonist ntawm chav kawm tsis-ergoline.

Cabergoline:

Cabergoline , muag nyob hauv hom tshuaj npe Dostinex ntawm lwm tus, yog cov tshuaj dopaminergic siv hauv kev kho cov qib siab ntawm prolactin, prolactinomas, Parkinson tus kab mob, thiab rau lwm yam cim. Nws yog noj ntawm qhov ncauj.

Apomorphine:

Apomorphine , muag nyob rau hauv lub npe lag luam Apokyn ntawm lwm tus, yog ib hom aporphine muaj kev ua si uas tsis yog xaiv dopamine agonist uas ua rau ob qho tib si D 2 -zoo li, thiab kom muaj ntau yam tsawg dua, D 1 -zoo li cov neeg txais . Nws kuj ua raws li qhov tsis haum ntawm 5-HT 2 thiab α-adrenergic receptors nrog siab siab. Kev sib xyaw ua ke yog keeb kwm morphine decomposition khoom tsim los ntawm kev kub nyoos morphine nrog cov concentrated acid, yog li ntawd - morphine cov cim tom qab. Rov qab rau nws lub npe, apomorphine tsis tshua muaj morphine lossis nws lub cev pob txha, tsis yog nws khi rau opioid receptors. Tus apo - tom ntej cuam tshuam txog nws yog morphine derivative ("[los ntawm morphine \").

Piribedil:

Piribedil (cov npe ua lag luam Pronoran , Trivastal Retard , Trastal , Trivastan , Clarium thiab lwm tus) yog tus sawv cev antiparkinsonian thiab piperazine derivative uas ua raws li D 2 thiab D 3 receptor agonist. Nws kuj muaj α 2 -adrenergic antagonist lub zog.

Rotigotine:

Rotigotine , muag nyob hauv hom npe nrov npe Neupro ntawm lwm tus, yog dopamine agonist ntawm chav tsis-ergoline cov tshuaj ntawm cov tshuaj tau qhia rau kev kho mob Parkinson tus kab mob (PD) thiab mob ceg tsis tswm (RLS). Nws yog tsim raws li kev hloov pauv ib zaug ib hnub twg uas muab cov tshuaj qeeb thiab tas li ntawm cov tshuaj dhau ntawm 24 teev.

ATC code N04:

ATC code N04 Cov tshuaj tiv thaiv cov tshuaj tiv thaiv kab mob yog kev siv tshuaj ntawm Anatomical Kev Ntsuas Tshuaj Classification System, ib qho kev hloov kho cov txheej txheem alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N04 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

Selegiline:

Selegiline , tseem hu ua L -deprenyl thiab muag hauv qab cov npe lag luam Eldepryl thiab Emsam ntawm lwm tus, yog cov tshuaj uas siv los kho tus kab mob Parkinson thiab muaj kev nyuaj siab tsis zoo. Nws tau muab nyob rau hauv daim ntawv ntawm tshuaj ntsiav los yog ntsiav tshuaj noj ntawm qhov ncauj rau Parkinson tus kab mob thiab ua ib thaj rau daim tawv nqaij rau kev nyuaj siab.

Rasagiline:

Rasagiline yog tshuaj tua tsis tau tus mob ntawm monoamine oxidase-B siv los ua kev kho mob los kho cov tsos mob thaum ntxov Parkinson tus kab mob los yog ua ib qho kev kho mob rau ntau yam mob.

ATC code N04:

ATC code N04 Cov tshuaj tiv thaiv cov tshuaj tiv thaiv kab mob yog kev siv tshuaj ntawm Anatomical Kev Ntsuas Tshuaj Classification System, ib qho kev hloov kho cov txheej txheem alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N04 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

Tolcapone:

Tolcapone , muag hauv cov lag luam muaj npe yog Tasmar , yog cov tshuaj siv los kho tus kab mob Parkinson (PD). Nws yog ib qho xaiv xaiv, muaj zog thiab thim rov qab nitrocatechol-hom inhibitor ntawm enzyme catechol- O -methyltransferase (COMT). Nws tau pom tias lub siab ua rau lub siab ua haujlwm tsis zoo, uas tau ua rau kev ncua ntawm kev tso cai ua lag luam hauv ntau lub tebchaws.

Entacapone:

Entacapone , muag nyob hauv cov lag luam muaj npe Comtan ntawm lwm tus, yog cov tshuaj siv feem ntau siv nrog lwm cov tshuaj rau kev kho mob ntawm Parkinson tus kab mob. Entacapone ua ke nrog levodopa thiab carbidopa tso cai levodopa kom muaj kev cuam tshuam ntev dua nyob rau hauv lub hlwb thiab txo qis cov kab mob Parkinson thiab cov tsos mob rau lub sijhawm ntev dua li levodopa thiab kho carbidopa ib leeg.

Budipine:

Budipine yog tus sawv cev antiparkinson ua lag luam rau kev kho mob ntawm tus kab mob Parkinson.

ATC code N05:

ATC code N05 Psycholeptics yog kev kho mob sib cais ntawm Anatomical Kev Ntsuas Cov Tshuaj Hauv Tshuaj, lub kaw lus ntawm cov cim alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N05 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

ATC code N05:

ATC code N05 Psycholeptics yog kev kho mob sib cais ntawm Anatomical Kev Ntsuas Cov Tshuaj Hauv Tshuaj, lub kaw lus ntawm cov cim alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N05 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

ATC code N05:

ATC code N05 Psycholeptics yog kev kho mob sib cais ntawm Anatomical Kev Ntsuas Cov Tshuaj Hauv Tshuaj, lub kaw lus ntawm cov cim alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N05 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

Chlorpromazine:

Chlorpromazine ( CPZ ), ua lag luam hauv qab cov npe lag luam Thorazine thiab Largactil ntawm lwm tus, yog cov tshuaj tiv thaiv kev tsis haum tshuaj. Nws yog feem ntau siv los kho cov kev puas siab puas ntsws xws li schizophrenia. Lwm yam kev siv suav nrog kev kho mob ntawm kev puas siab puas ntsws bipolar, kev coj tus cwj pwm tsis zoo hauv cov menyuam yaus suav nrog kev saib xyuas kev tsis txaus siab, xeev siab thiab ntuav, ntxhov siab ua ntej kev phais mob, thiab hiccups uas tsis txhim kho raws li lwm cov kev ntsuas. Nws tuaj yeem muab los ntawm qhov ncauj, los ntawm kev txhaj tshuaj rau hauv cov leeg, lossis mus rau txoj hlab ntshav.

Levomepromazine:

Levomepromazine , tseem hu ua methotrimeprazine , yog ib qho tshuaj phenothiazine neuroleptic. Hom tshuaj npe suav nrog Nozinan, Levoprome, Detenler, Hirnamin, Levotomin thiab Neurocil. Nws yog qhov muaj zog qis-tawm tsam kev tiv thaiv kom muaj zog analgesic, hypnotic thiab antiemetic zog uas feem ntau siv hauv kev saib xyuas palliative.

Promazine:

Promazine yog cov tshuaj uas yog rau cov chav kawm phenothiazine ntawm tshuaj tiv thaiv kev puas hlwb. Cov tshuaj qub siv los kho tus mob schizophrenia, nws tseem raug kho, nrog rau cov neeg sawv cev tshiab xws li olanzapine thiab quetiapine. Nws muaj feem ntau anticholinergic phiv, tab sis yog extrapyramidal kev phiv tsis yooj yim dua yog. Nws yooj yim dissolves hauv cawv.

Acepromazine:

Acepromazine , acetopromazine, lossis acetylpromazine yog phenothiazine derivative tshuaj tiv thaiv kev tsis haum tshuaj. Nws tau siv nyob rau hauv tib neeg thaum lub sijhawm xyoo 1950 yog kev tawm tsam, tab sis tam sim no yuav luag tshwj xeeb siv rau ntawm cov tsiaj ua sedative thiab antiemetic. Nws muaj feem xyuam nrog tshuaj analogue, chlorpromazine, tseem tseem siv ua tshuaj tiv thaiv kabmob hauv tib neeg. Acepromazine feem ntau yog siv tshuaj los kho hauv kev tua tsiaj los yog txhav tsiaj.

Triflupromazine:

Triflupromazine ( Vesprin ) yog cov tshuaj tiv thaiv kev ntxhov siab ntawm chav kawm phenothiazine. Ntawm cov teebmeem sib txawv ntawm kev qhia txog triflupromazine rau kev siv cov tshuaj no yog emesis hnyav thiab Hiccups hnyav. Vim nws cov peev xwm phiv nws tsis yog kub tus qauv hauv kev kho mob tiv thaiv kab mob.

Cyamemazine:

Cyamemazine ( Tercian ), tseem hu ua cyamepromazine , yog cov tshuaj tiv thaiv kev tiv thaiv tsis zoo ntawm chav kawm phenothiazine uas tau qhia los ntawm Theraplix hauv Fabkis xyoo 1972 thiab tom qab ntawd hauv Portugal zoo li.

Chlorproethazine:

Chlorproethazine , muag nyob rau hauv cov npe lag luam tshuaj Neuriplege , yog ib cov tshuaj ntawm phenothiazine pawg tau piav qhia tias yog cov leeg ua kom cov leeg ua kom lub cev tsis zoo lossis ua kom lub cev tsis zoo uas yog lossis tau ua lag luam nyob hauv Europe raws li cov tshuaj pleev rau kev kho mob leeg. Nws tau cuam tshuam nrog photoallergic contact dermatitis.

ATC code N05:

ATC code N05 Psycholeptics yog kev kho mob sib cais ntawm Anatomical Kev Ntsuas Cov Tshuaj Hauv Tshuaj, lub kaw lus ntawm cov cim alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N05 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

Dixyrazine:

Dixyrazine , tseem hu ua dixypazin (oxalate), muag hauv qab hom npe Ansiolene , Esocalm , Esucos , Metronal , thiab Roscal , yog ib cov tshuaj tiv thaiv kev pheej hmoo ntawm phenothiazine pab pawg tau piav raws li neuroleptic thiab antihistamine. Nws tau xub pib qhia nyob rau hauv lub teb chaws Yelemees xyoo 1969. Nws yog siv los ua tus mob neuroleptic, anxiolytic, thiab tshuaj antihistamine nyob rau hauv cov koob tshuaj 12,5 txog 75 mg rau ib hnub.

Fluphenazine:

Fluphenazine , muag nyob hauv cov npe lag luam Prolixin ntawm lwm tus, yog cov tshuaj tiv thaiv kev puas hlwb. Nws yog siv nyob rau hauv kev kho mob ntawm kev puas siab ntsws xws li mob schizophrenia, thiab zoo li muaj qhov sib npaug hauv kev ua tau zoo rau qhov qis-potency antipsychotics zoo li chlorpromazine. Nws yog muab los ntawm qhov ncauj, txhaj rau hauv cov leeg, lossis hauv qab daim tawv. Kuj tseem muaj qhov ua yeeb yaj kiab ntev ntev uas siv tau ntev txog plaub asthiv. Fluphenazine decanoate, daim ntawv txhaj tshuaj rau cov tshuaj fluphenazine, yuav tsum tsis txhob siv los ntawm cov neeg muaj kev nyuaj siab heev.

Perphenazine:

Perphenazine yog ib qho tshuaj tiv thaiv kev tsis raug. Chemically, nws tau muab cais raws li cov tshuaj piperazinyl phenothiazine. Ameslikas lag luam hauv Asmeskas raws li Trilafon, nws tau nyob hauv kev siv tshuaj rau ntau xyoo lawm.

Prochlorperazine:

Prochlorperazine , yav dhau los muag nyob rau hauv cov npe kws muaj npe Compazine ntawm lwm tus, yog cov tshuaj siv los kho mob xeev siab, mob schizophrenia, migraines, thiab ntxhov siab. Nws yog qhov siv tshuaj tsawg dua rau qhov kev ntxhov siab. Nws tuaj yeem noj los ntawm qhov ncauj, kho qhov quav, txhaj rau hauv leeg ntshav, lossis txhaj tshuaj rau hauv cov leeg.

Thiopropazate:

Thiopropazate yog cov tshuaj tiv thaiv kev tiv thaiv tsis zoo ntawm chav kawm phenothiazine. Nws yog cov khoom prodrug rau perphenazine.

Trifluoperazine:

Trifluoperazine , muag nyob rau hauv ntau tus naj npawb ntawm cov npe lag luam, yog ib qho kev tiv thaiv kev tiv thaiv ib txwm siv los kho tus mob schizophrenia Nws kuj tseem siv tau lub sijhawm luv luv hauv cov neeg uas muaj kev ntxhov siab dav dav tab sis tsis tshua nyiam benzodiazepines. Nws yog ntawm chav kawm phenothiazine tshuaj lom neeg.

Acetophenazine:

Acetophenazine ( Tindal ) yog cov tshuaj tiv thaiv kev tiv thaiv tsis haum ntawm chav kawm phenothiazine.

Thioproperazine:

Thioproperazine , muag nyob rau hauv lub npe hom Majeptil , yog ib qho kev tiv thaiv tsis haum ntawm phenothiazine pawg uas yog siv los ua tus mob plab, antiemetic, sedative, thiab hauv kev kho mob schizophrenia thiab manic theem ntawm kev puas siab puas ntsws bipolar. Majeptil muaj nyob hauv 10 mg ntsiav tshuaj.

Butaperazine:

Butaperazine yog cov tshuaj tiv thaiv kev tiv thaiv tawm tsam phenothiazine chav kawm.

Perazine:

Perazine ( Taxilan ) yog ib nrab-potency ntse antipsychotic ntawm chav kawm phenothiazine. Nws yog qhov zoo heev rau chlorpromazine, thiab ua raws li dopamine antagonist. Xyoo 2014 kev tshuaj xyuas zoo sib piv nws nrog lwm cov tshuaj tiv thaiv kev ntxhov siab:

ATC code N05:

ATC code N05 Psycholeptics yog kev kho mob sib cais ntawm Anatomical Kev Ntsuas Cov Tshuaj Hauv Tshuaj, lub kaw lus ntawm cov cim alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N05 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

Periciazine:

Periciazine (INN), tseem hu ua pericyazine (BAN) lossis propericiazine , yog ib cov tshuaj uas yog rau phenothiazine chav kawm ntawm cov tshuaj tiv thaiv kev tiv thaiv ib txwm muaj.

Thioridazine:

Thioridazine yog thawj lub tshuaj tiv thaiv kev tiv thaiv kab mob los ntawm pab pawg phenothiazine thiab yav dhau los tau siv dav hauv kev kho mob schizophrenia thiab psychosis. Cov khoom muaj npe tau raug rho tawm thoob ntiaj teb xyoo 2005 vim tias nws ua rau mob plawv dhia tsis xwm yeem. Txawm li cas los xij, cov qauv kho cov tseem muaj nyob hauv Asmeskas.

Mesoridazine:

Mesoridazine (Serentil) yog piperidine neuroleptic siv rau cov tshuaj hauv chav kawm hu ua phenothiazines, siv nyob rau hauv kev kho mob schizophrenia. Nws yog cov tshuaj metabolite ntawm thioridazine. Lub npe tshuaj tau muab los ntawm kuv thyl s ulf o xy thiab cov yeeb nkab tshem tawm cov pawg ua haujlwm hauv nws cov qauv tshuaj.

Pipotiazine:

Pipotiazine ( Piportil ), tseem hu ua pipothiazine , yog cov tshuaj tiv thaiv kev tiv thaiv ntawm chav kawm phenothiazine uas tau siv hauv tebchaws Askiv thiab lwm lub tebchaws rau kev kho mob schizophrenia. Nws cov khoom zoo ib yam li cov tshuaj chlorpromazine. Xyoo 2004 kev tshuaj xyuas tau tshawb xyuas nws qhov ua tau zoo rau cov neeg muaj tus mob schizophrenia:

ATC code N05:

ATC code N05 Psycholeptics yog kev kho mob sib cais ntawm Anatomical Kev Ntsuas Cov Tshuaj Hauv Tshuaj, lub kaw lus ntawm cov cim alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N05 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

Haloperidol:

Haloperidol , muag nyob hauv hom lag luam npe Haldol ntawm lwm tus, yog ib hom tshuaj tiv thaiv kev tsis haum tshuaj. Haloperidol yog siv rau kev kho mob schizophrenia, tics hauv Tourette syndrome, mania hauv kev puas siab puas ntsws bipolar, delirium, ntxhov siab, mob hlwb, thiab mob hlwb hauv kev thim kev haus cawv. Tej zaum nws yuav siv los ntawm qhov ncauj lossis txhaj tshuaj rau hauv cov leeg lossis leeg ntshav. Haloperidol feem ntau ua haujlwm tsis pub dhau 30 mus rau 60 feeb. Kev tsim qauv ntev ntev yuav raug siv los ua kev txhaj tshuaj txhua plaub lub lis piam rau cov neeg muaj tus mob schizophrenia lossis mob lwm yam mob, uas tsis nco qab lossis tsis kam noj tshuaj ntawm qhov ncauj.

Trifluperidol:

Trifluperidol yog cov tshuaj tiv thaiv kev tawm tsam tsis zoo ntawm cov tshuaj butyrophenone. Nws muaj cov khoom dav dav zoo ib yam li cov ntawm haloperidol, tab sis yog qhov muaj txiaj ntsig ntau los ntawm qhov hnyav, thiab ua rau muaj kev phiv ntau dua, tshwj xeeb tshaj yog kev tuaj yeem ua rau dyskinesia thiab lwm yam kev cuam tshuam ntxiv. Nws yog siv nyob rau hauv kev kho mob ntawm lub hlwb xws li mania thiab schizophrenia. Nws tau tshwm sim ntawm Janssen Pharmaceutica hauv 1959.

Melperone:

Melperone yog atypical antipsychotic ntawm chav kawm butyrophenone chemical, ua rau nws muaj kev cuam tshuam txog cov tshuaj tiv thaiv kev pheej hmoo haloperidol. Nws thawj zaug nkag mus rau kev siv tshuaj rau xyoo 1960.

Moperone:

Moperone yog cov tshuaj tiv thaiv kev ntxhov siab ntawm chav kawm butyrophenone.

Pipamperone:

Pipamperone , tseem hu ua carpiperone thiab floropipamide lossis fluoropipamide , thiab raws li floropipamide hydrochloride (JAN), yog ib qho kev tiv thaiv kabmob ntawm tsev neeg butyrophenone siv rau kev kho mob schizophrenia thiab ua kev pabcuam tsaug zog rau kev nyuaj siab. Nws yog lossis tau ua lag luam nyob hauv cov npe lag luam nrog rau Dipiperon , Dipiperal , Piperonil , Piperonyl , thiab Propitan . Pipamperone nrhiav tau ntawm Janssen Pharmaceutica hauv xyoo 1961, thiab nkag mus hauv cov chaw kuaj mob hauv Tebchaws Asmeskas xyoo 1963.

Bromperidol:

Bromperidol yog butyrophenone derivative. Nws yog ib qho muaj zog thiab ntev ntev kev coj ntawm neuroleptic, siv los ua tshuaj tiv thaiv kev kho mob ntawm tus mob schizophrenia. Nws tau tshwm sim ntawm Janssen Pharmaceutica hauv xyoo 1966.

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Benperidol:

Benperidol , muag nyob rau hauv lub npe lag luam Anquil ntawm lwm tus, yog tshuaj uas yog qhov muaj txiaj ntsig zoo butyrophenone derivative. Nws yog cov neuroleptic muaj zog tshaj plaws nyob rau hauv European kev ua lag luam, nrog chlorpromazine kev sib txig sib luag li 75 txog 100. Nws yog cov tshuaj tiv thaiv kab mob, uas tuaj yeem siv rau kev kho mob schizophrenia, tab sis feem ntau yog siv los tswj hypersexuality syndromes thiab qee zaum sau rau cov neeg ua txhaum kev sib daj sib deev raws li muaj kev sib deev, ua lwm txoj hauv kev los tiv thaiv tshuaj androgen xws li cyproterone acetate.

Droperidol:

Droperidol yog ib qho tshuaj antidopaminergic siv raws li antiemetic thiab ua tshuaj tiv thaiv kab mob. Droperidol feem ntau kuj tseem siv tau ua sedative hauv kev kho mob hnyav.

Fluanisone:

Fluanisone yog ib txwm muaj tshuaj tiv thaiv kev ntxhov siab thiab ua kom loog ntawm butyrophenone chemical chav kawm. Nws yog siv nyob rau hauv kev kho mob ntawm schizophrenia thiab mania. Nws tseem yog qhov tseem ceeb ntawm cov ntawv txhaj tshuaj tiv thaiv kab mob hauv fentanyl / fluanisone (Hypnorm) qhov twg nws yog siv rau kev ua nas nyob ua haujlwm thaum lub sijhawm ua haujlwm luv.

Azaperone:

Azaperone yog pyridinylpiperazine thiab butyrophenone neuroleptic tshuaj nrog sedative thiab antiemetic cuam tshuam, uas yog siv ua feem ntau yog siv tshuaj tranquilizer hauv veterinary tshuaj. Nws yog qhov tsis tshua muaj siv nyob rau hauv tib neeg raws li tshuaj tiv thaiv kev puas tsuaj.

ATC code N05:

ATC code N05 Psycholeptics yog kev kho mob sib cais ntawm Anatomical Kev Ntsuas Cov Tshuaj Hauv Tshuaj, lub kaw lus ntawm cov cim alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N05 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

Oxypertine:

Oxypertine yog tshuaj tiv thaiv kev kho mob uas siv los kho tus mob schizophrenia. Nws tseem tau raug soj ntsuam los kho kev ntxhov siab ntawm kev noj tshuaj ntau npaum li 20 mg rau ib hnub. Chemically, nws yog ib qho indole thiab phenylpiperazine derivative. Zoo li reserpine thiab tetrabenazine, oxygenpertine depletes catecholamines, txawm hais tias tsis serotonin, muaj peev xwm pom nws qhov kev ua tau zoo ntawm neuroleptic. Nws cov qauv zoo ib yam li Solypertine thiab milipertine.

Molindone:

Molindone , muag nyob rau hauv cov npe muaj npe Moban , yog cov tshuaj tiv thaiv kev puas hlwb uas yog siv hauv Tebchaws Asmeskas hauv kev kho mob schizophrenia. Nws ua haujlwm los ntawm kev thaiv cov teebmeem ntawm dopamine hauv hlwb, uas ua rau cov tsos mob ploj zuj zus ntawm lub hlwb. Nws yog nqus sai sai thaum coj qhov ncauj.

Sertindole:

Sertindole , muag nyob hauv hom tshuaj npe Serdolect ntawm lwm tus, yog tshuaj tiv thaiv kev puas hlwb. Sertindole tau tsim los ntawm lub tuam txhab ua lag luam Danish Lundbeck thiab tau txais kev lag luam hauv kev tso cai los ntawm Abbott Labs. Zoo li lwm yam atypical antipsychotics, nws muaj kev ua si ntawm dopamine thiab serotonin receptors hauv lub hlwb. Nws yog siv nyob rau hauv kev kho mob ntawm schizophrenia. Nws yog cais cov tshuaj raws li phenylindole derivative.

Ziprasidone:

Ziprasidone , muag nyob hauv hom tshuaj npe Geodon ntawm lwm tus, yog atypical antipsychotic siv los kho tus mob schizophrenia thiab kev puas siab puas ntsws bipolar. Nws yuav raug siv los ntawm qhov ncauj thiab los ntawm kev txhaj tshuaj rau hauv cov leeg (IM). Daim foos IM siv tau rau kev ntxhov siab mob hnyav hauv cov neeg muaj tus mob schizophrenia.

Lurasidone:

Lurasidone , muag nyob hauv kev lag luam tawm lub npe Latuda ntawm lwm tus, yog cov tshuaj tiv thaiv kev puas tsuaj uas siv los kho tus mob schizophrenia thiab kev puas siab puas ntsws bipolar. Hauv kev bipolar nws yuav siv nrog ua ke nrog kev siab ntsiag to xws li lithium lossis valproate. Nws yog noj ntawm qhov ncauj.

ATC code N05:

ATC code N05 Psycholeptics yog kev kho mob sib cais ntawm Anatomical Kev Ntsuas Cov Tshuaj Hauv Tshuaj, lub kaw lus ntawm cov cim alphanumeric tsim los ntawm World Health Organization (WHO) rau kev faib tawm cov tshuaj thiab lwm cov khoom kho mob. Pawg N05 yog ib feem ntawm cov pab pawg anatomical N Cov kab mob tsis zoo .

Flupentixol:

Flupentixol (INN), tseem hu ua flupenthixol , ua lag luam hauv qab cov npe lag luam xws li Depixol thiab Fluanxol yog cov tshuaj tiv thaiv kev pheej hmoo ntawm cov thioxanthene chav kawm. Nws tau qhia hauv xyoo 1965 los ntawm Lundbeck. Ntxiv rau kev npaj tshuaj ib leeg, nws kuj tseem muaj xws li flupentixol / melitracen - cov khoom sib txuam uas muaj ob qho tib si melitracen thiab flupentixol.nFlupentixol tsis pom zoo rau siv hauv Tebchaws Asmeskas. Nws yog, txawm li cas los xij, kev pom zoo rau kev siv nyob rau hauv UK, Australia, Canada, Lavxias Federation, South Africa, New Zealand, Philippines thiab ntau lub tebchaws.

Clopenthixol:

Clopenthixol ( Sordinol ), tseem hu ua clopentixol , yog ib qho tshuaj tiv thaiv kev tsis haum tshuaj ntawm thioxanthene chav kawm. Nws tau qhia los ntawm Lundbeck xyoo 1961.

Chlorprothixene:

Chlorprothixene , muag nyob rau hauv hom lag luam npe Truxal ntawm lwm tus, yog ib qho kev tiv thaiv kom tsis haum ntawm thioxanthene pawg.

Tiotixene:

Tiotixene , lossis thiothixene , muag hauv qab cov npe lag luam Navane ntawm lwm tus, yog cov tshuaj tiv thaiv kev tiv thaiv tsis zoo ntawm chav thioxanthene uas cuam tshuam nrog chlorprothixene thiab yog siv rau hauv kev kho mob hlwb xws li schizophrenia thiab bipolar mania. Nws tau tsim tawm hauv Tebchaws Asmeskas xyoo 1967 los ntawm Pfizer.

Zuclopenthixol:

Zuclopenthixol , tseem hu ua zuclopentixol , yog ib hom tshuaj siv los kho tus mob schizophrenia thiab lwm yam kev mob hlwb. Nws yog classed, pharmacologically, raws li ib txwm tiv thaiv tshuaj tiv thaiv. Chemically nws yog thioxanthene. Nws yog cis -isomer ntawm clopenthixol. Clopenthixol tau qhia rau xyoo 1961, thaum zuclopenthixol tau qhia rau xyoo 1978.

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